What is Cyclobenzaprine used for? (Cyclobenzaprine para que sirve?)
The drug is designed to quickly relieve muscle cramps. It relaxes the muscles and helps cope with myalgia without directly affecting the muscular frame. The active ingredient of the drug is cyclobenzaprine. It is an effective myotropic antispasmodic that works regardless of the cause of muscle pain. It has been well studied and is recognized as safe for patients over 18 years of age.
Cyclobenzaprine is more than 90% bound to plasma albumin and globulin. Its bioavailability ranges from 33 to 55%. Maximum blood concentration is reached 8 hours after oral administration.
Cyclobenzaprine affects brain stem cells. The active substance partially interferes with the transmission of nerve impulses from the CNS to the periphery and restructures the spinal cord. This provides a relaxing effect.
When using the drug Yuredol, tonic activity is reduced; spasms, cramps, tremors are eliminated; a sedative effect is provided.
Hypertonicity and pain under the influence of cyclobenzaprine disappear. At the same time, there is no effect on the very muscular frame and synapses. In spasticity against the background of cerebral palsy, the drug is ineffective, but it can be used as a concomitant therapy for tetanus.
How should Cyclobenzaprine 10 mg be used correctly? (Cyclobenzaprine 10 mg para que sirve)
The drug can be used as an independent remedy and as part of complex therapy. It comes in the form of tablets for oral administration. The concentration of the active component is 10 mg. This is enough to relieve muscle cramps and improve well-being. The effectiveness of Yuredol tablets can be increased by physical therapy methods.
Drugs with cyclobenzaprine in the composition are prescribed for regular smooth muscle cramps, regardless of the cause. Yuredol can improve the quality of life of a patient suffering from acute or chronic pain, but the effectiveness and duration of use may vary from case to case. The pills can also be used in the recovery period after surgery. The drug promotes faster rehabilitation after joint surgery. Another indication for the use of Cyclobenzaprine in a dosage of 10 mg is recovery from injuries. The active ingredient will help to reduce pain for bruises, sprains, cracked bones, dislocations, fractures.
There is no universal scheme for taking the tablets. The daily dose and duration of the therapeutic course are always determined by the attending physician, taking into account the indications and the initial state of the patient. The drug can be taken regardless of food. Studies have shown that eating increases the bioavailability of the active component, but this indicator does not affect the effectiveness of therapy.
The minimum daily dose is one tablet. It’s possible to increase the concentration if the effect of treatment is insignificant. The course of intake shouldn’t exceed 2-4 weeks. If you take the drug less than the specified period, painful sensations and hypertonicity of smooth muscles will return. If the permissible duration is exceeded, the risk of developing tolerance to cyclobenzaprine increases. Maximum benefit is registered on the seventh day from the beginning of therapy.
According to the instructions, Yuredol tablets should not be taken if there are contraindications. The main restrictions are:
history of myocardial infarction;
hyperfunction of the thyroid gland;
pathology of the pituitary gland;
age under 18 years old.
Cyclobenzaprine-based muscle relaxants should not be combined with alcoholic beverages and several drugs. The combination of monoamine oxidase inhibitors and CNS stimulants is especially dangerous. Ignoring this requirement is fraught with the development of intoxication. Symptoms of poisoning - nausea, vomiting, tachycardia, dizziness, hallucinations. In severe cases, confusion, blockage of the respiratory center, coma, and death are possible.
Patients who have prescribed tablets with cyclobenzaprine in the composition are warned about possible side effects. Prolonged intake may provoke:
The risk of side effects is higher if you are prone to allergic reactions and elderly. If the symptoms do not worsen the quality of life and pass on their own after a while, there is no need for treatment. In case of pronounced side effects, correction of the therapeutic dose or prescription of another muscle relaxant is necessary.
Violation of the instructions and independent increase in the recommended dosage may cause intoxication. In severe overdose, hypotension, seizures, tachycardia, and somnolence develop. In critical cases, cardiac arrest is possible, as well as death.
The treatment in case of overdose is gastric lavage and taking sorbents if you remain conscious. Heart rate and blood pressure should also be monitored. In case of arrhythmia, intravenous administration of alkaline solutions is indicated. Seizures are controlled with benzodiazepines.
How long does Cyclobenzaprine last?
The effect of taking the pills comes quickly. The first positive changes are noticeable after 2-3 hours. They intensify during the next 5-6 hours. Within 7-9 hours after taking, the muscle pain will be weak. Hypertonicity will not bother the patient.
If the next dose of the drug is not taken, the effect weakens. Within 1.5 days, the active ingredient is eliminated. Cyclobenzaprine is metabolized in the kidneys. It is excreted from the body in the form of glucuronides.
It’s not recommended to interrupt the course of treatment earlier than the term specified by the doctor. After discontinuation of the drug after 2-4 weeks of treatment, the patient's well-being remains stable. Muscle pain and increased smooth muscle tone do not bother.